SCHEMBL9804896

SCHEMBL9804896

CCC(C#N)(Cc1cncnc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.37
CYP19A1 P11511 5/20 0.37
EBP Q15125 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
CCR1 P32246 1/20 0.34
CTSL P07711 1/20 0.34
CYP2D6 P10635 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
OPRM1 P35372 1/20 0.33
DRD3 P35462 1/20 0.33
LMNA P02545 1/20 0.33
KCNA5 P22460 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10625675 0.84 ATM (0.47) ATMEBPSIGMAR1CYP1A2CYP3A4
SCHEMBL9804836 0.82 EBP (0.41) ATMCYP19A1EBPSIGMAR1CYP1A2
SCHEMBL9804729 0.81 CYP19A1 (0.52) ATMCYP19A1CYP3A4CCR1
SCHEMBL9804855 0.79 EBP (0.41) ATMCYP19A1EBPSIGMAR1CYP3A4
SCHEMBL9805022 0.78 CYP19A1 (0.59) ATMCYP19A1CYP3A4
SCHEMBL13271382 0.78 CYP2D6 (0.44) ATMEBPSIGMAR1CYP3A4CYP2C19
SCHEMBL9804889 0.78 CYP1A2 (0.37) ATMEBPSIGMAR1CYP1A2CYP3A4
SCHEMBL9804705 0.77 CYP19A1 (0.39) CYP19A1EBPSIGMAR1
SCHEMBL9804866 0.77 CYP19A1 (0.45) ATMCYP19A1EBPSIGMAR1CYP3A4
SCHEMBL9804741 0.77 CYP19A1 (0.34) ATMCYP19A1EBPSIGMAR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed