SCHEMBL9804855

SCHEMBL9804855

CCCCC(C#N)(Cc1cncnc1)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EBP Q15125 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CYP19A1 P11511 4/20 0.35
ATM Q13315 2/20 0.35
EPHB4 P54760 1/20 0.33
TEK Q02763 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
CTSL P07711 2/20 0.32
CTSS P25774 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
HSD11B1 P28845 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CNR2 P34972 2/20 0.31
CNR1 P21554 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804907 0.85 CYP19A1 (0.43) EBPSIGMAR1CYP19A1CYP3A4
SCHEMBL9804675 0.82 CYP2C9 (0.39) EBPSIGMAR1CYP19A1HDAC1CTSL
SCHEMBL10371783 0.81 CYP3A4 (0.44) EBPSIGMAR1CYP19A1CTSLCTSS
SCHEMBL9804896 0.79 ATM (0.37) EBPSIGMAR1CYP19A1ATMCTSL
SCHEMBL9804705 0.77 CYP19A1 (0.39) EBPSIGMAR1CYP19A1CYP11B1CYP11B2
SCHEMBL9804836 0.77 EBP (0.41) EBPSIGMAR1CYP19A1ATMCTSL
SCHEMBL9804684 0.76 EBP (0.33) EBPSIGMAR1CNR2CNR1
SCHEMBL10372958 0.75 TDP1 (0.43) EBPSIGMAR1CYP3A4CYP2D6CYP2C9
SCHEMBL51900 0.73 EBP (0.59) EBPSIGMAR1ATMCYP3A4CYP2D6
SCHEMBL9805022 0.73 CYP19A1 (0.59) CYP19A1ATMCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed