SCHEMBL9809336

SCHEMBL9809336

O=C(N1CCOCC1)N1CCN(CCCOc2ccc(F)cc2)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.66
HRH2 P25021 2/20 0.66
HRH3 Q9Y5N1 6/20 0.60
FKBP1A P62942 1/20 0.59
LMNA P02545 2/20 0.56
HTR2A P28223 3/20 0.56
SIGMAR1 Q99720 2/20 0.56
HTR1A P08908 2/20 0.56
DRD2 P14416 2/20 0.56
DRD3 P35462 2/20 0.56
TMEM97 Q5BJF2 1/20 0.56
ALDH1A1 P00352 2/20 0.56
MAPK1 P28482 2/20 0.56
CYP1A2 P05177 1/20 0.56
CHRM2 P08172 1/20 0.56
CHRM1 P11229 1/20 0.56
SCN1A P35498 1/20 0.56
HTR2B P41595 1/20 0.56
KCNH2 Q12809 1/20 0.56
SCN2A Q99250 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9809294 0.88 HRH1 (0.64) HRH1HRH2HRH3LMNAHTR2A
SCHEMBL9809263 0.87 USP2 (0.72) HRH1HRH2HRH3LMNAHTR2A
SCHEMBL9809418 0.87 HRH3 (0.64) HRH1HRH2HRH3LMNAHTR2A
SCHEMBL9809235 0.86 HRH1 (0.63) HRH1HRH2HRH3LMNAHTR2A
SCHEMBL9809346 0.84 HRH1 (0.57) HRH1HRH2HRH3LMNAHTR2A
SCHEMBL9809405 0.83 HRH3 (0.61) HRH1HRH2HRH3LMNASIGMAR1
SCHEMBL3586381 0.82 HRH3 (0.66) HRH1HRH2HRH3HTR2ASIGMAR1
SCHEMBL9809297 0.82 HRH1 (0.63) HRH1HRH2HRH3LMNAHTR2A
SCHEMBL1728918 0.81 USP2 (0.78) HRH1HRH2HRH3LMNAHTR2A
SCHEMBL9809231 0.79 HRH1 (0.63) HRH1HRH2HRH3LMNAHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0211928-B1 PIPERAZINECARBOXAMIDES HAVING A PHENOXYALKYL OR THIOPHENOXYALKYL SIDE CHAIN AB LEO (SE) 1991-05-02 EP claimed
US-4778789-A PSYCHOLOGICAL DISORDERS AKTIEBOLAGET LEO (SE) 1988-10-18 US claimed
EP-0211928-B1 PIPERAZINECARBOXAMIDES HAVING A PHENOXYALKYL OR THIOPHENOXYALKYL SIDE CHAIN AB LEO (SE) 1991-05-02 EP disclosed
US-4778789-A PSYCHOLOGICAL DISORDERS AKTIEBOLAGET LEO (SE) 1988-10-18 US disclosed