SCHEMBL9809443

SCHEMBL9809443

CCOC(=O)C1=C(CCC(O)c2ccccc2)NC(C)=C(C(=O)OC)C1c1ccccc1SC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.49
CACNA1C Q13936 4/20 0.49
TBXA2R P21731 3/20 0.49
ADRA1A P35348 3/20 0.49
SLC6A3 Q01959 3/20 0.49
HTR1A P08908 2/20 0.49
ADRA2A P08913 2/20 0.49
CHRM1 P11229 2/20 0.49
DRD1 P21728 2/20 0.49
SLC6A2 P23975 2/20 0.49
OPRM1 P35372 2/20 0.49
DRD3 P35462 2/20 0.49
KCNH2 Q12809 2/20 0.49
ABCB11 O95342 2/20 0.49
ABCB1 P08183 2/20 0.49
ADRB3 P13945 2/20 0.49
OPRK1 P41145 2/20 0.49
SCN5A Q14524 2/20 0.49
KCNK2 O95069 1/20 0.49
ADRB2 P07550 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426346 0.96 CACNA1C (0.47) ADORA3CACNA1CTBXA2RADRA1ASLC6A3
SCHEMBL10615427 0.84 ADORA3 (0.52) ADORA3CACNA1CTBXA2RADRA1ASLC6A3
SCHEMBL7467067 0.84 CACNA1C (0.51) ADORA3CACNA1CTBXA2RADRA1ASLC6A3
SCHEMBL7435874 0.83 ADORA3 (0.54) ADORA3CACNA1CCYP2C9CYP3A4MEN1
SCHEMBL10614837 0.83 TBXA2R (0.58) ADORA3CACNA1CTBXA2RADRA1ASLC6A3
SCHEMBL7275805 0.83 TBXA2R (0.57) ADORA3CACNA1CTBXA2RADRA1ASLC6A3
SCHEMBL7268196 0.83 ADORA3 (0.52) ADORA3CACNA1CTBXA2RADRA1ASLC6A3
SCHEMBL7467069 0.81 ADORA3 (0.50) ADORA3CACNA1CTBXA2RADRA1ASLC6A3
SCHEMBL7437789 0.80 CACNA1D (0.55) ADORA3CACNA1CADRA1ADRD1OPRM1
SCHEMBL7428216 0.80 CACNA1B (0.58) ADORA3CACNA1CTBXA2RADRA1ASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5075324-A ARALKYL-1,4-DIHYDROPYRIDINES, A METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1991-12-24 US disclosed