SCHEMBL9809458

SCHEMBL9809458

CCN(C)CC#CCCC(=O)C(O)(c1ccccc1)C1CCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 6/20 0.51
CHRM2 P08172 3/20 0.51
CHRM1 P11229 3/20 0.51
CYP2C19 P33261 2/20 0.51
KCNH2 Q12809 2/20 0.51
SLC6A3 Q01959 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
PKM P14618 1/20 0.51
NFKB1 P19838 1/20 0.51
THPO P40225 1/20 0.51
ABCB11 O95342 1/20 0.51
ESR1 P03372 1/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51
ADRA2A P08913 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
TBXA2R P21731 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9809560 0.98 CHRM3 (0.53) CHRM3CHRM2CHRM1CYP2C19KCNH2
SCHEMBL9809558 0.97 CHRM3 (0.55) CHRM3CHRM2CHRM1CYP2C19KCNH2
Water SCHEMBL9618799 0.96 CHRM3 (0.54) CHRM3CHRM2CHRM1CYP2C19KCNH2
SCHEMBL9809462 0.95 CHRM3 (0.47) CHRM3CHRM2CHRM1CYP2C19KCNH2
SCHEMBL7650415 0.92 CHRM3 (0.51) CHRM3CHRM2CHRM1CYP2C19KCNH2
Hydrochloric Acid SCHEMBL9809457 0.91 MEN1 (0.52) CHRM3CHRM2CHRM1CYP2C19KCNH2
SCHEMBL9618849 0.90 ALDH1A1 (0.54) CHRM3CHRM2CHRM1CYP2C19KCNH2
SCHEMBL9809464 0.88 CHRM3 (0.55) CHRM3CHRM2CHRM1CYP2C19KCNH2
SCHEMBL9809567 0.88 CHRM3 (0.55) CHRM3CHRM2CHRM1CYP2C19KCNH2
SCHEMBL7913118 0.88 CHRM3 (0.55) CHRM3CHRM2CHRM1CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5036107-A Treatment of neurogenic bladder disorders MARION MERRELL DOW INC. (US) 1991-07-30 US disclosed
EP-0414180-A2 Hydroxylated ene ketones, acetylenic grignards and hydroxylated yne ketones therefrom MARION MERRELL DOW INC. (US) 1991-02-27 EP disclosed
US-4973756-A Hydroxylated ene ketones, acetylenic grignards and hydroxylated yne ketones therefrom MARION LABORATORIES, INC. (US) 1990-11-27 US disclosed