SCHEMBL9810221

SCHEMBL9810221

CC(=O)Oc1ccc(SC2CCCc3cccnc32)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.38
SLC6A3 Q01959 2/20 0.38
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ABCB11 O95342 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADRA2A P08913 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
PDE4A P27815 1/20 0.38
ADRA1A P35348 1/20 0.38
OPRK1 P41145 1/20 0.38
STAT6 P42226 1/20 0.38
HIF1A Q16665 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
PDPK1 O15530 1/20 0.35
PGR P06401 1/20 0.35
CHRM2 P08172 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10571311 0.99 ESR1 (0.37) ESR1SLC6A3LMNAKDM4EABCB11
SCHEMBL9810223 0.84 DDB1 (0.44) PDPK1ADORA2ACXCR4
Hydrochloric Acid SCHEMBL10571722 0.83 DDB1 (0.43) PDPK1ADORA2ACXCR4
SCHEMBL9810224 0.82 DDB1 (0.39) KDM4ECXCR4KMT2AALDH1A1MAPT
Hydrochloric Acid SCHEMBL10570078 0.81 DDB1 (0.38) KDM4ECXCR4KMT2AALDH1A1MAPT
SCHEMBL10574015 0.81 DDB1 (0.46) KDM4EHDAC1HDAC6CXCR4KMT2A
Hydrochloric Acid SCHEMBL10569604 0.81 HDAC1 (0.43) KDM4EHDAC1HDAC6ADORA2ACXCR4
SCHEMBL9810216 0.81 CYP2D6 (0.39) CYP3A4CYP2C9CXCR4KMT2AMAPT
SCHEMBL9810209 0.80 CXCR4 (0.40) HDAC1HDAC6CXCR4
SCHEMBL9810195 0.80 DDB1 (0.40) CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254611-B1 DERIVATIVES OF 8-PHENYLTHIOTETRAHYDROQUINOLINES AND THEIR SALTS, THEIR SYNTHESIS FOR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1991-06-12 EP disclosed
EP-0254611-A1 Derivatives of 8-phenylthiotetrahydroquinolines and their salts, their synthesis for use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1988-01-27 EP disclosed