SCHEMBL9810223

SCHEMBL9810223

COc1ccc(SC2CCCc3cccnc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44
PDPK1 O15530 1/20 0.40
CXCR4 P61073 12/20 0.40
CYP2D6 P10635 2/20 0.37
ADORA2A P29274 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10571722 0.99 DDB1 (0.43) DDB1CRBNPDPK1CXCR4CYP2D6
SCHEMBL9810224 0.88 DDB1 (0.39) DDB1CRBNCXCR4CYP2D6
Hydrochloric Acid SCHEMBL10570078 0.86 DDB1 (0.38) DDB1CRBNCXCR4CYP2D6
SCHEMBL9810216 0.85 CYP2D6 (0.39) DDB1CRBNCXCR4CYP2D6
SCHEMBL9810195 0.85 DDB1 (0.40) DDB1CRBNCXCR4CYP2D6
SCHEMBL9810221 0.84 ESR1 (0.38) PDPK1CXCR4ADORA2A
Hydrochloric Acid SCHEMBL10568508 0.84 TAOK1 (0.38) DDB1CRBNCXCR4CYP2D6
Hydrochloric Acid SCHEMBL10569209 0.84 CXCR4 (0.40) DDB1CRBNCXCR4CYP2D6
SCHEMBL9770476 0.84 HTR6 (0.40) DDB1CRBNCXCR4CYP2D6
Hydrochloric Acid SCHEMBL10571311 0.83 ESR1 (0.37) PDPK1CXCR4ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254611-B1 DERIVATIVES OF 8-PHENYLTHIOTETRAHYDROQUINOLINES AND THEIR SALTS, THEIR SYNTHESIS FOR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1991-06-12 EP disclosed
EP-0254611-A1 Derivatives of 8-phenylthiotetrahydroquinolines and their salts, their synthesis for use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1988-01-27 EP disclosed