SCHEMBL9811910

SCHEMBL9811910

O=C(Nc1ccccc1)C(P(=O)(O)O)P(=O)(O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.55
CA12 O43570 1/20 0.52
CA9 Q16790 1/20 0.52
MAPT P10636 4/20 0.50
ALDH1A1 P00352 4/20 0.50
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
GAA P10253 2/20 0.50
ATM Q13315 2/20 0.50
TP53 P04637 1/20 0.50
EPHX1 P07099 1/20 0.50
TSHR P16473 1/20 0.50
EPHX2 P34913 1/20 0.50
CDK9 P50750 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
LMNA P02545 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9811837 0.81 NPC1 (0.50) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL9811900 0.81 CA12 (0.55) POLBCA12MAPTALDH1A1MEN1
SCHEMBL9338142 0.81 ALDH1A1 (0.56) POLBCA12CA9MAPTALDH1A1
SCHEMBL233680 0.78 CA9 (0.50) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL9811890 0.77 HTT (0.58) ALDH1A1MEN1KMT2ASMN1; SMN2GAA
SCHEMBL9811846 0.77 CA12 (0.58) CA12ALDH1A1SMN1; SMN2TP53EPHX2
SCHEMBL11882145 0.74 POLB (0.63) POLBMAPTALDH1A1MEN1KMT2A
SCHEMBL21056246 0.73 MEN1 (0.61) POLBMAPTALDH1A1MEN1KMT2A
SCHEMBL11758471 0.73 MAPT (0.61) POLBMAPTALDH1A1MEN1KMT2A
SCHEMBL10623171 0.73 CA9 (0.58) CA12CA9MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0243173-B1 NEW DIPHOSPHONIC ACID COMPOUNDS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-06-26 EP disclosed
US-4963536-A INHIBIT BONE RESORPTION FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1990-10-16 US disclosed
US-4857513-A Diphosphonic acid compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISIWA PHARMACEUTICAL CO., LTD. (JP) 1989-08-15 US disclosed
EP-0243173-A2 New diphosphonic acid compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-10-28 EP disclosed
US-4124371-A α,α-DIPHOSPHONATO ACETANILIDES MONSANTO COMPANY (US) 1978-11-07 US disclosed
US-4124371-A α,α-DIPHOSPHONATO ACETANILIDES MONSANTO COMPANY (US) 1978-11-07 US disclosed
US-3906062-A Alpha,alpha-diphosphonato acetanilides MONSANTO CO 1975-09-16 US disclosed
US-3906062-A Alpha,alpha-diphosphonato acetanilides MONSANTO CO 1975-09-16 US disclosed