SCHEMBL9813945

SCHEMBL9813945

C[C@H](Cc1ccc(O)cc1)N(CC(O)c1cccc(Br)c1)CC(O)c1cccc(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.40
SLC6A2 P23975 2/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
ADRB2 P07550 7/20 0.39
OPRM1 P35372 4/20 0.39
CYP3A4 P08684 3/20 0.39
MAPK1 P28482 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
HIF1A Q16665 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ADRB1 P08588 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADRB3 P13945 1/20 0.39
PTGS1 P23219 1/20 0.39
HTR2A P28223 1/20 0.39
SLC6A4 P31645 1/20 0.39
MC4R P32245 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9813952 0.85 SLC2A1 (0.50) ADRB2CYP3A4CYP2D6HIF1AADRB1
SCHEMBL9813921 0.85 MAOB (0.42) TAAR1SLC6A2ESR1ESR2ADRB2
SCHEMBL9813912 0.85 MAOB (0.42) TAAR1SLC6A2ESR1ESR2ADRB2
SCHEMBL9813875 0.85 SLC2A1 (0.50) ADRB2CYP3A4CYP2D6HIF1AADRB1
SCHEMBL9813982 0.85 SLC2A1 (0.50) ADRB2CYP3A4CYP2D6HIF1AADRB1
SCHEMBL9813872 0.85 SLC2A1 (0.50) ADRB2CYP3A4CYP2D6HIF1AADRB1
SCHEMBL9813944 0.85 SLC2A1 (0.50) ADRB2CYP3A4CYP2D6HIF1AADRB1
SCHEMBL9813900 0.85 SLC2A1 (0.50) ADRB2CYP3A4CYP2D6HIF1AADRB1
SCHEMBL9813936 0.84 AOC3 (0.47) TAAR1SLC6A2ESR1ESR2OPRM1
SCHEMBL9813928 0.84 AOC3 (0.47) TAAR1SLC6A2ESR1ESR2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017619-A Anitdiabetic HOFFMANN-LA ROCHE INC. (US) 1991-05-21 US disclosed
EP-0198412-B1 PHENETHANOL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1989-03-22 EP disclosed