SCHEMBL9814027

SCHEMBL9814027

C[C@H](Cc1ccc(O)cc1)N(CC(O)c1ccccc1)CC(O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.47
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
OPRK1 P41145 8/20 0.44
OPRM1 P35372 7/20 0.44
OPRD1 P41143 7/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TAAR1 Q96RJ0 2/20 0.42
SLC6A2 P23975 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9813936 1.00 AOC3 (0.47) AOC3ESR1ESR2OPRK1OPRM1
SCHEMBL9814024 1.00 AOC3 (0.47) AOC3ESR1ESR2OPRK1OPRM1
SCHEMBL9813943 1.00 AOC3 (0.47) AOC3ESR1ESR2OPRK1OPRM1
SCHEMBL9813928 1.00 AOC3 (0.47) AOC3ESR1ESR2OPRK1OPRM1
SCHEMBL9813937 0.89 SLC2A1 (0.47)
SCHEMBL9813948 0.89 SLC2A1 (0.47)
SCHEMBL11021733 0.87 AOC3 (0.46) AOC3OPRK1KDM4EMEN1KMT2A
SCHEMBL9813944 0.84 SLC2A1 (0.50)
SCHEMBL9813900 0.84 SLC2A1 (0.50)
SCHEMBL9813952 0.84 SLC2A1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017619-A Anitdiabetic HOFFMANN-LA ROCHE INC. (US) 1991-05-21 US disclosed
EP-0198412-B1 PHENETHANOL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1989-03-22 EP disclosed
EP-0198412-A1 Phenethanol amine derivatives F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1986-10-22 EP disclosed