SCHEMBL9814124

SCHEMBL9814124

COc1cc2c(cc1O)C(C1=NCCN1)CCC2

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.53
ADRA2A P08913 3/20 0.53
CYP2D6 P10635 2/20 0.53
HTR1A P08908 1/20 0.53
OPRM1 P35372 1/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
ALDH1A1 P00352 1/20 0.52
BLM P54132 1/20 0.52
TAAR1 Q96RJ0 1/20 0.52
MAOA P21397 2/20 0.48
DRD1 P21728 1/20 0.46
DRD5 P21918 1/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10749519 0.99 CYP2D6 (0.54) ADRA1AADRA2ACYP2D6HTR1AOPRM1
SCHEMBL9814120 0.95 ADRA1A (0.53) ADRA1AADRA2ACYP2D6HTR1AOPRM1
Hydrochloric Acid SCHEMBL10749333 0.94 CYP2D6 (0.54) ADRA1AADRA2ACYP2D6HTR1AOPRM1
Hydrochloric Acid SCHEMBL10749865 0.89 CYP2D6 (0.59) ADRA1AADRA2ACYP2D6HTR1AOPRM1
SCHEMBL768674 0.86 ADRA1A (0.62) ADRA1AADRA2ACYP2D6HTR1AOPRM1
SCHEMBL2776285 0.84 ADRA1A (0.54) ADRA1AADRA2ACYP2D6HTR1AOPRM1
SCHEMBL769213 0.78 CYP2D6 (0.62) ADRA1AADRA2ACYP2D6HTR1AOPRM1
SCHEMBL769130 0.78 ADRA1A (0.62) ADRA1AADRA2ACYP2D6HTR1AOPRM1
Hydrochloric Acid SCHEMBL10751218 0.77 CYP2D6 (0.63) ADRA1AADRA2ACYP2D6HTR1AOPRM1
Hydrochloric Acid SCHEMBL10749411 0.77 CYP2D6 (0.63) ADRA1AADRA2ACYP2D6HTR1AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0166937-B1 ADRENERGIC COMPOUNDS ABBOTT LABORATORIES (US) 1991-08-28 EP disclosed