SCHEMBL9815840

SCHEMBL9815840

Cc1cncc(C(=O)N(NC(=O)c2ccc([N+](=O)[O-])cc2)C(C)(C)C)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 6/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 1/20 0.46
POLB P06746 1/20 0.46
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9425631 0.96 ABCB1 (0.48) ABCB1CYP3A4CYP2C9POLBHPGD
SCHEMBL9714538 0.84 POLB (0.63) ABCB1CYP3A4CYP2C9POLBHPGD
SCHEMBL8166763 0.80 POLB (0.74) ABCB1CYP3A4CYP2C9POLBHPGD
SCHEMBL9652010 0.80 POLB (0.74) ABCB1CYP3A4CYP2C9POLBHPGD
SCHEMBL9495409 0.76 ABCB1 (0.60) ABCB1CYP3A4CYP2C9POLBHPGD
SCHEMBL9714310 0.74 POLB (0.68) ABCB1CYP3A4CYP2C9POLB
SCHEMBL25381850 0.73 CYP11B1 (0.64) POLBSMN1; SMN2NPC1RAB9A
SCHEMBL30354874 0.73 CYP11B1 (0.64) POLBSMN1; SMN2NPC1RAB9A
SCHEMBL9714603 0.73 CYP3A4 (0.73) ABCB1CYP3A4CYP2C9POLB
SCHEMBL5057049 0.73 ABCB1 (0.78) ABCB1CYP3A4CYP2C9POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed