SCHEMBL9816822

SCHEMBL9816822

CC(N)=CC(=O)NC(C)C

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
MMP1 P03956 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34
CA9 Q16790 1/20 0.34
LMNA P02545 1/20 0.32
ALOX15 P16050 1/20 0.32
BLM P54132 1/20 0.32
PMP22 Q01453 1/20 0.32
OPRK1 P41145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9816818 1.00 TSHR (0.50) TSHRALDH1A1GAACA12CA1
SCHEMBL13174451 0.80 TSHR (0.54) TSHRALDH1A1GAACA12CA1
SCHEMBL16365865 0.79 TSHR (0.48) TSHRALDH1A1GAACA12CA1
SCHEMBL21160229 0.78 ALDH1A1 (0.54) TSHRALDH1A1GAACA12CA1
SCHEMBL16532707 0.76 TSHR (0.50) TSHRALDH1A1GAACA12CA1
SCHEMBL13174334 0.76 TSHR (0.50) TSHRALDH1A1GAACA12CA1
SCHEMBL16000934 0.76 TSHR (0.50) TSHRALDH1A1GAACA12CA1
SCHEMBL16532709 0.76 TSHR (0.50) TSHRALDH1A1GAACA12CA1
SCHEMBL16532708 0.75 TSHR (0.54) TSHRALDH1A1GAACA12CA1
SCHEMBL27840741 0.74 ALDH1A1 (0.50) TSHRALDH1A1GAACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220653-B1 3-AMINOCARBONYL-1,4-DIHYDROPYRIDINE-5-CARBOXYLIC ACID COMPOUNDS, PROCESS FOR PREPARATION AND USE THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Nippon Shoji Kabushiki Kaisha (JP) 1991-11-06 EP disclosed
US-4874773-A HYPOTENSIVE AGENTS, VASODILATORS NIPPON SHOJI KABUSHIKI KAISHA (JP) 1989-10-17 US disclosed
EP-0220653-A2 3-Aminocarbonyl-1,4-dihydropyridine-5-carboxylic acid compounds, process for preparation and use thereof, and pharmaceutical composition containing the same Nippon Shoji Kabushiki Kaisha (JP) 1987-05-06 EP disclosed