SCHEMBL9817849

SCHEMBL9817849

CCOC(=O)CCCCc1ccc(C#Cc2ccc3c(c2)C(C)(C)CCS3)cc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.58
RARG P13631 10/20 0.58
RARA P10276 9/20 0.58
CYP3A4 P08684 3/20 0.58
KMT2A Q03164 1/20 0.58
CYP26A1 O43174 2/20 0.48
CYP4Z1 Q86W10 2/20 0.40
RXRA P19793 2/20 0.38
CRABP2 P29373 1/20 0.37
CYP4F11 Q9HBI6 1/20 0.36
CYP4F12 Q9HCS2 1/20 0.36
CYP4F2 P78329 2/20 0.36
CYP4A11 Q02928 2/20 0.36
ALOX5 P09917 1/20 0.35
FFAR1 O14842 1/20 0.34
ACACB O00763 1/20 0.34
SSTR5 P35346 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817673 0.97 RARB (0.58) RARBRARGRARACYP3A4KMT2A
SCHEMBL9817773 0.92 RARA (0.55) RARBRARGRARACYP3A4KMT2A
SCHEMBL8674175 0.90 CYP3A4 (0.46) RARBRARGRARACYP3A4KMT2A
SCHEMBL6671541 0.90 RARA (0.70) RARBRARGRARACYP3A4KMT2A
SCHEMBL9817641 0.89 RARA (0.56) RARBRARGRARACYP3A4KMT2A
SCHEMBL6665899 0.88 RARB (0.62) RARBRARGRARACYP3A4KMT2A
SCHEMBL6668823 0.87 RARB (0.53) RARBRARGRARACYP3A4KMT2A
SCHEMBL6668880 0.86 RARB (0.54) RARBRARGRARACYP3A4KMT2A
SCHEMBL9817631 0.86 RARA (0.54) RARBRARGRARACYP3A4KMT2A
SCHEMBL6664870 0.86 RARB (0.62) RARBRARGRARACYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed