SCHEMBL9821858

SCHEMBL9821858

COC(=O)C1CCc2ccc(O)cc2O1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.51
ESR2 Q92731 1/20 0.51
CHRNA7 P36544 1/20 0.47
DRD2 P14416 1/20 0.46
DRD1 P21728 1/20 0.46
DRD4 P21917 1/20 0.46
DRD5 P21918 1/20 0.46
DRD3 P35462 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29052788 0.89 CYP4F2 (0.53) ESR1ESR2
SCHEMBL23360606 0.85 GABRA1 (0.46) ESR1ESR2
SCHEMBL9837746 0.85 CYP4F2 (0.62) ESR1ESR2DRD2DRD1DRD4
SCHEMBL9838425 0.85 CYP4F2 (0.62) ESR1ESR2DRD2DRD1DRD4
SCHEMBL1019684 0.85 CYP4F2 (0.62) ESR1ESR2DRD2DRD1DRD4
SCHEMBL29586758 0.85 CYP4F2 (0.62) ESR1ESR2DRD2DRD1DRD4
SCHEMBL9838132 0.82 ESR1 (0.56) ESR1ESR2DRD2DRD1DRD4
SCHEMBL7111420 0.82 ESR1 (0.56) ESR1ESR2DRD2DRD1DRD4
SCHEMBL7111422 0.82 ESR1 (0.56) ESR1ESR2DRD2DRD1DRD4
SCHEMBL24496703 0.81 ESR1 (0.52) ESR1ESR2DRD2DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292977-B1 ALKOXY-SUBSTITUTED DIHYDROBENZOPYRAN-2-CARBOXYLATE DERIVATIVES G.D. Searle & Co. (US) 1991-09-04 EP disclosed
US-4889871-A ANTIINFLAMMATORY AGENTS; SELECTIVE LEUKOTRIENE ANTAGONISTS G. D. SEARLE & CO. (US) 1989-12-26 US disclosed
EP-0292977-A1 Alkoxy-substituted dihydrobenzopyran-2-carboxylate derivatives G.D. Searle & Co. (US) 1988-11-30 EP disclosed