SCHEMBL9821873

SCHEMBL9821873

COc1ccc(CN(C)Cc2cccc3ccccc23)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.68
CYP1A2 P05177 2/20 0.68
CYP2C19 P33261 2/20 0.68
ACHE P22303 2/20 0.66
NR1I2 O75469 2/20 0.66
LMNA P02545 2/20 0.66
SLC6A2 P23975 2/20 0.66
HTR2A P28223 2/20 0.66
SLC6A4 P31645 2/20 0.66
KCNH2 Q12809 2/20 0.66
SIGMAR1 Q99720 2/20 0.66
ADRA2A P08913 1/20 0.66
KMT2A Q03164 5/20 0.64
MEN1 O00255 4/20 0.64
L3MBTL1 Q9Y468 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
SMPD1 P17405 1/20 0.50
PTPN1 P18031 1/20 0.50
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9695219 0.90 ACHE (0.70) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL10484897 0.83 CYP2D6 (0.60) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL9721972 0.83 CYP2D6 (0.74) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL9858161 0.83 CYP2D6 (0.74) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL10932466 0.82 CYP2D6 (1.00) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL9722081 0.82 CYP2D6 (0.72) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL3243955 0.82 CYP2D6 (0.72) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL9722034 0.82 CYP2D6 (0.72) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL9722021 0.82 CYP2D6 (0.72) CYP2D6CYP1A2CYP2C19ACHENR1I2
SCHEMBL29336388 0.81 CYP1A2 (0.56) CYP2D6CYP1A2CYP2C19LMNASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221781-B1 BENZYLAMINE DERIVATIVES, PROCESS FOR PRODUCTION THEREOF, AND USE THEREOF MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-05-02 EP disclosed
US-4822822-A FUNGICIDES FOR PLANTS AND ANIMALS MITSUI TOATSU CHEMICALS, INC. (JP) 1989-04-18 US disclosed
EP-0221781-A2 Benzylamine derivatives, process for production thereof, and use thereof MITSUI TOATSU CHEMICALS, Inc. (JP) 1987-05-13 EP disclosed