SCHEMBL9822639

SCHEMBL9822639

CCCC(C)OC(=O)C1=C(C)NC(Cn2ccnc2)=C(C(=O)O)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
CYP1A2 P05177 4/20 0.49
CYP3A4 P08684 4/20 0.49
CYP2C9 P11712 4/20 0.49
CYP2C19 P33261 4/20 0.49
LMNA P02545 3/20 0.49
MAPT P10636 3/20 0.49
CYP2D6 P10635 2/20 0.49
TSHR P16473 2/20 0.49
NFKB1 P19838 2/20 0.49
THPO P40225 2/20 0.49
CACNA1C Q13936 8/20 0.49
CACNA1F O60840 7/20 0.49
CACNA1D Q01668 7/20 0.49
CACNA1S Q13698 7/20 0.49
ADORA3 P0DMS8 3/20 0.49
NR1I2 O75469 2/20 0.48
AGTR1 P30556 2/20 0.48
PDE4D Q08499 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9766585 0.88 CACNA1F (0.51) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9787339 0.85 CACNA1F (0.62) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9787471 0.84 HIF1A (0.57) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9787403 0.84 CACNA1F (0.68) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9787465 0.83 HIF1A (0.62) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9787472 0.79 CACNA1F (0.57) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9787287 0.79 MEN1 (0.61) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL10663251 0.79 CACNA1B (0.49) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL10663093 0.79 CACNA1B (0.49) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL10756245 0.79 CACNA1C (0.60) MEN1KMT2ACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0172029-B1 1,4-DIHYDROPYRIDINES JOHN WYETH & BROTHER LIMITED (GB) 1991-02-27 EP claimed
CN-85106495-A The method for preparing heterogeneous ring compound 1987-02-11 CN claimed
EP-0172029-A1 1,4-Dihydropyridines JOHN WYETH & BROTHER LIMITED (GB) 1986-02-19 EP claimed