SCHEMBL9823461

SCHEMBL9823461

C#CCN(Cc1ccc2nc[nH]c(=O)c2c1)c1cc(OC)c(OC)c(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 1.00
TYMS P04818 6/20 0.50
IP6K1 Q92551 2/20 0.43
IP6K3 Q96PC2 1/20 0.42
IP6K2 Q9UHH9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823440 0.83 DHFR (0.70) DHFRTYMS
SCHEMBL18163434 0.81 DHFR (0.78) DHFRTYMS
SCHEMBL9823134 0.79 DHFR (1.00) DHFRTYMS
SCHEMBL9823448 0.79 DHFR (0.69) DHFRTYMS
SCHEMBL9823110 0.78 DHFR (0.79) DHFRTYMS
SCHEMBL9823189 0.77 DHFR (0.61) DHFRTYMS
SCHEMBL9823212 0.70 DHFR (0.50) DHFRTYMS
SCHEMBL9247891 0.70 DHFR (0.68) DHFR
SCHEMBL9255306 0.69 DHFR (0.63) DHFR
SCHEMBL9253629 0.69 NAMPT (0.73) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP claimed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US claimed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP claimed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO claimed
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed