SCHEMBL9823943

SCHEMBL9823943

CC(C)(Cc1ccc(Cl)c(C(F)(F)F)c1)C(=O)CBr

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.46
KDR P35968 1/20 0.42
PYCR1 P32322 1/20 0.42
P2RX7 Q99572 6/20 0.41
AURKA O14965 1/20 0.40
RPS6KB1 P23443 1/20 0.40
AURKB Q96GD4 1/20 0.40
ABCB11 O95342 1/20 0.40
KDM4E B2RXH2 1/20 0.39
FAAH O00519 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
GPR84 Q9NQS5 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
PDK1 Q15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823633 0.80 EPHX1 (0.43) PPARGPPARA
SCHEMBL2600033 0.77 IDO1 (0.57) IDO1KDRPYCR1P2RX7LMNA
SCHEMBL9200306 0.76 GSK3B (0.50) LMNAPPARA
SCHEMBL9380085 0.76 SLC6A4 (0.48) LMNAMAPTPPARGPPARA
SCHEMBL1720743 0.74 IDO1 (0.58) IDO1KDRPYCR1P2RX7LMNA
SCHEMBL31731921 0.73 IDO1 (0.61) IDO1KDRPYCR1P2RX7ABCB11
SCHEMBL120051 0.73 IDO1 (0.61) IDO1KDRPYCR1P2RX7ABCB11
SCHEMBL1590516 0.71 RXRA (0.55) IDO1KDRP2RX7ABCB11FAAH
SCHEMBL30302148 0.71 RXRA (0.55) IDO1KDRP2RX7ABCB11FAAH
SCHEMBL11434970 0.71 IDO1 (0.54) IDO1KDRPYCR1P2RX7ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301393-B1 1,4-DISUBSTITUTED 1-AZOLYL-3,3-DYMETHYLBUTANE DERIVATIVES BAYER AG (DE) 1991-08-14 EP disclosed
EP-0301393-A1 1,4-Disubstituted 1-azolyl-3,3-dymethylbutane derivatives BAYER AG (DE) 1989-02-01 EP disclosed