SCHEMBL9824152

SCHEMBL9824152

CCn1c2cc(N3CCN(C)CC3)c(F)cc2c(=O)c2c(=O)[nH]sc21

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.50
GAA P10253 1/20 0.48
RAD52 P43351 1/20 0.48
KDM4E B2RXH2 6/20 0.46
ALDH1A1 P00352 4/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
NPC1 O15118 1/20 0.46
HPGD P15428 1/20 0.46
POLB P06746 1/20 0.45
GLA P06280 1/20 0.44
ALK Q9UM73 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2933050 0.90 KDM4E (0.48) DRD3KDM4EALDH1A1HPGD
SCHEMBL609448 0.90 ALDH1A1 (0.52) DRD3KDM4EALDH1A1HPGD
SCHEMBL605962 0.88 KDM4E (0.41) DRD3GAARAD52KDM4EALDH1A1
SCHEMBL8921044 0.83 GAA (0.43) DRD3GAARAD52KDM4EALDH1A1
SCHEMBL9824069 0.83 KDM4E (0.41) KDM4EALDH1A1HPGD
SCHEMBL9824093 0.83 PRKD3 (0.47)
SCHEMBL607251 0.82
SCHEMBL10188340 0.82 KCNH2 (0.43)
SCHEMBL2936532 0.82 KCNH2 (0.43)
SCHEMBL9214098 0.81 KDM4E (0.45) KDM4EALDH1A1HPGDALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed