SCHEMBL9824329

SCHEMBL9824329

NC1CCN(c2c(F)cc3c(=O)c4c(=O)[nH]oc4n(C4CC4)c3c2Br)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
PIM1 P11309 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
PIM3 Q86V86 1/20 0.41
CSNK1G1 Q9HCP0 1/20 0.41
TOP2A P11388 13/20 0.40
TOP2B Q02880 10/20 0.40
TOP1 P11387 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9825282 0.90 PIM1 (0.50) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824606 0.89 ALDH1A1 (0.55) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL10667865 0.85 PIM1 (0.46) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824506 0.85 ALDH1A1 (0.38) ALDH1A1POLBOPRM1TOP2ATOP2B
SCHEMBL9824228 0.82 IKBKB (0.50) PIM1GSK3A
SCHEMBL9824074 0.81 KMT2A (0.46) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9825057 0.81 PRKD3 (0.48) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9837629 0.79 PIM1 (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL9839219 0.78 PIM1 (0.44) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824649 0.78 PIM1 (0.45) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed