SCHEMBL9824464

SCHEMBL9824464

CCOC(=O)c1c(SC)n(-c2ccncc2)c2c(F)c(F)c(F)cc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
STAT3 P40763 2/20 0.42
HTT P42858 1/20 0.38
ALDH1A1 P00352 5/20 0.36
NPSR1 Q6W5P4 4/20 0.36
HPGD P15428 4/20 0.36
MAPT P10636 2/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
HSD17B10 Q99714 3/20 0.35
ALOX15 P16050 2/20 0.35
KDM5A P29375 1/20 0.35
KDM5B Q9UGL1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824642 0.90 MEN1 (0.41) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824142 0.90 MEN1 (0.46) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824444 0.90 ALDH1A1 (0.47) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824403 0.89 MEN1 (0.45) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824566 0.87 PDE4D (0.44) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824453 0.87 KMT2A (0.45) MEN1KMT2AALDH1A1NPSR1HPGD
SCHEMBL9824276 0.85 RXFP1 (0.38) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824260 0.84 MEN1 (0.41) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824799 0.83 STAT3 (0.38) MEN1KMT2ASTAT3HTTALDH1A1
SCHEMBL9824691 0.83 MEN1 (0.42) MEN1KMT2AHTTALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed