Bromide

Bromide

SCHEMBL9826548

CCOC(=O)c1ccc(C[P+](c2ccccc2)(c2ccccc2)c2ccccc2)cc1Cl.[Br-]

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.47
CYP4A11 Q02928 1/20 0.47
TSHR P16473 3/20 0.45
BAZ2B Q9UIF8 1/20 0.41
BAZ2A Q9UIF9 1/20 0.41
ALDH1A1 P00352 4/20 0.40
HSD17B10 Q99714 2/20 0.40
SNCA P37840 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
MAPT P10636 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
TNF P01375 1/20 0.39
LMNA P02545 1/20 0.39
HSP90AA1 P07900 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8651071 0.87 SNCA (0.42) TSHRALDH1A1HSD17B10SNCAMAPT
Bromide SCHEMBL9827145 0.84 TSHR (0.44) TSHRALDH1A1MAPTKDM4EHPGD
SCHEMBL10003354 0.79 CYP4F2 (0.60) CYP4F2CYP4A11TSHRBAZ2BBAZ2A
Bromide SCHEMBL9826440 0.79 SMN1; SMN2 (0.58) ALDH1A1SNCACA12CA1CA2
Bromide SCHEMBL7025256 0.78 CYP4F2 (0.56) CYP4F2CYP4A11ALDH1A1SNCACA2
SCHEMBL522636 0.77 CYP4F2 (0.57) CYP4F2CYP4A11TSHRBAZ2BBAZ2A
Bromide SCHEMBL3918746 0.76 TSHR (0.57) TSHRALDH1A1HSD17B10KDM4ETDP1
Bromide SCHEMBL21176866 0.76 L3MBTL1 (0.47) TSHRALDH1A1MAPTHPGDLMNA
SCHEMBL20077738 0.76 SMN1; SMN2 (0.57) CYP4F2CYP4A11TSHRBAZ2BBAZ2A
SCHEMBL6971203 0.76 CYP4F2 (0.78) CYP4F2CYP4A11TSHRBAZ2BBAZ2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0150892-B1 SUBSTITUTED ALKYLIDENE IMIDAZOLES G.D. Searle & Co. (US) 1991-04-24 EP disclosed
US-4837333-A SELECTIVE INHIBITOR OF THROMBOXANE SYNTHETASE ENZYME G. D. SEARLE & CO. (US) 1989-06-06 US disclosed
EP-0150892-A2 Substituted alkylidene imidazoles G.D. Searle & Co. (US) 1985-08-07 EP disclosed