SCHEMBL9827449

SCHEMBL9827449

CN(C)C1CCN2C(=O)OCc3cccc1c32

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.44
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
KCNH2 Q12809 1/20 0.38
HTR6 P50406 6/20 0.37
ACHE P22303 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828644 0.84 HTR1A (0.41) HTR1AHTR6
SCHEMBL9827759 0.80 HTR1A (0.41) HTR1AHTR6
SCHEMBL9828705 0.80 HTR1A (0.41) HTR1ASLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL9828460 0.79 HTR1A (0.42) HTR1AHTR6
SCHEMBL9828411 0.71 HTR1A (0.42) HTR1A
SCHEMBL7376163 0.70 HTR1A (0.73) HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL10658365 0.68 CES1 (0.51) HTR1A
SCHEMBL9827478 0.66 CES1 (0.42) HTR1AHTR6
SCHEMBL9830196 0.64 MAP2K1 (0.41) HTR1AHTR6
SCHEMBL11719507 0.63 HTR1A (0.40) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0239129-B1 HYDROQUINOLINE COMPOUNDS, COMPOSITIONS CONTAINING SAME AND PROCESSES FOR PREPARING SAME OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-09-25 EP disclosed
US-4963566-A ANTIULCER AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-10-16 US disclosed
EP-0239129-A2 Hydroquinoline compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-09-30 EP disclosed