SCHEMBL9831111

SCHEMBL9831111

CC1C(=O)Nc2cc(N)c([N+](=O)[O-])cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.48
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
TSHR P16473 2/20 0.39
MAPT P10636 9/20 0.38
TDP1 Q9NUW8 5/20 0.38
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 3/20 0.38
POLB P06746 3/20 0.38
KMT2A Q03164 3/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
MCL1 Q07820 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GALR3 O60755 1/20 0.37
THRB P10828 1/20 0.37
MPI P34949 1/20 0.36
LMNA P02545 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833104 0.94 PGR (0.48) PGRCYP1A2CYP2C9CYP2C19TSHR
SCHEMBL9833325 0.84 CYP1A2 (0.41) PGRCYP1A2CYP2C9CYP2C19TSHR
SCHEMBL9834197 0.81 CYP1A2 (0.39) CYP1A2CYP2C9CYP2C19TSHRMAPT
SCHEMBL9832370 0.81 PGR (0.40) PGRCYP1A2CYP2C9CYP2C19TSHR
SCHEMBL9834174 0.80 CYP1A2 (0.38) CYP1A2CYP2C9CYP2C19TSHRMAPT
SCHEMBL10470349 0.79 MAPT (0.40) CYP1A2CYP2C9CYP2C19TSHRMAPT
Hydrochloric Acid SCHEMBL10374033 0.79 PGR (0.43) PGR
SCHEMBL9833951 0.78 CYP1A2 (0.37) CYP1A2CYP2C9CYP2C19TSHRMAPT
SCHEMBL9832943 0.78 MAPT (0.39) CYP1A2CYP2C9CYP2C19TSHRMAPT
SCHEMBL9832383 0.78 CYP1A2 (0.41) PGRCYP1A2CYP2C9CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
CN-85103724-B Process for preparing pyrrolobenzimidazoles 曼海姆伯灵格股份公司 1988-07-06 CN disclosed
CN-85103724-A The method for preparing novel pyrrolo-benzoglyoxaline 1986-07-02 CN disclosed