SCHEMBL9831503

SCHEMBL9831503

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2cccc(C(F)(F)F)c2)c2c1CSc1ccccc1-2

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
LMNA P02545 2/20 0.38
HTT P42858 1/20 0.38
NPY5R Q15761 3/20 0.37
TP53 P04637 2/20 0.37
KCNJ6 P48051 2/20 0.37
KCNJ5 P48544 2/20 0.37
KCNJ3 P48549 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KLKB1 P03952 1/20 0.36
POLB P06746 2/20 0.36
KMT2A Q03164 1/20 0.36
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831600 0.95 NPY5R (0.43) IDO1PTGS1PTGS2LMNAHTT
SCHEMBL9316246 0.95 IDO1 (0.44) IDO1PTGS1PTGS2LMNATP53
SCHEMBL9833522 0.90 TP53 (0.40) PTGS1PTGS2TP53KCNJ6KCNJ5
SCHEMBL8111901 0.90 TP53 (0.42) PTGS1PTGS2TP53KMT2A
SCHEMBL9831507 0.89 TP53 (0.44) PTGS1PTGS2TP53POLBCTSK
SCHEMBL9832082 0.89 MAPT (0.39) TP53POLB
SCHEMBL9833424 0.88 TP53 (0.38) TP53POLBKMT2A
SCHEMBL9832014 0.88 POLB (0.44) LMNATP53POLBKMT2A
SCHEMBL9833720 0.88 TP53 (0.38) PTGS1PTGS2TP53POLBKMT2A
SCHEMBL9834138 0.87 TP53 (0.42) TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed