SCHEMBL9832837

SCHEMBL9832837

COC(=O)C1(C)C(=O)Nc2cc3[nH]c(-c4cccnc4)nc3cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
HPGD P15428 3/20 0.50
HSD17B10 Q99714 1/20 0.50
MAPT P10636 5/20 0.49
KDM4E B2RXH2 4/20 0.49
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
STAT1 P42224 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
TP53 P04637 4/20 0.45
HTT P42858 1/20 0.44
CYP11B1 P15538 1/20 0.44
POLB P06746 2/20 0.43
KIT P10721 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833616 0.90 MAPT (0.47) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL9834034 0.89 ALDH1A1 (0.53) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL9830018 0.88 MAPT (0.51) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL9832543 0.88 PDE4A (0.62) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL10470322 0.87 ALDH1A1 (0.49) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL11025322 0.85 PDE4A (0.56) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL9830260 0.79 MAPT (0.46) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL9831255 0.79 MAPT (0.52) ALDH1A1HPGDHSD17B10MAPTKDM4E
SCHEMBL9834487 0.79 PDE4A (0.37) MAPTKDM4EPDE4APDE4BPDE4C
SCHEMBL9832117 0.79 MAPT (0.54) ALDH1A1HPGDHSD17B10MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed