SCHEMBL9833191

SCHEMBL9833191

CC1(C)C(=O)Nc2cc3[nH]c(C=Cc4ccncc4)nc3cc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.58
PDE4B Q07343 1/20 0.58
PDE4C Q08493 1/20 0.58
PDE4D Q08499 1/20 0.58
PDE3B Q13370 1/20 0.58
PDE3A Q14432 1/20 0.58
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43
RAB9A P51151 5/20 0.43
NPC1 O15118 4/20 0.43
MEN1 O00255 6/20 0.41
KMT2A Q03164 6/20 0.41
LMNA P02545 4/20 0.41
MAPT P10636 8/20 0.40
KDM4E B2RXH2 3/20 0.40
MCL1 Q07820 2/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
ATM Q13315 1/20 0.40
HTT P42858 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10477800 0.89 NPC1 (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834489 0.83 PDE3B (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834485 0.83 PDE3B (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10373985 0.81 ALDH1A1 (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834055 0.80 PDE3B (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834059 0.80 PDE3B (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9832377 0.79 PDE3B (0.50) PDE4APDE4BPDE4CPDE4DPDE3B
Adibendan SCHEMBL9832050 0.78 PDE3B (0.90) PDE4APDE4BPDE4CPDE4DPDE3B
Adibendan SCHEMBL10470994 0.77 PDE3B (0.88) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833827 0.77 PDE3B (0.48) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed