SCHEMBL9833592

SCHEMBL9833592

Fc1ccc(C2OC(=S)OC2(Cn2cncn2)c2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.46
CYP2C9 P11712 3/20 0.46
THRB P10828 1/20 0.45
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 2/20 0.36
NR1I2 O75469 1/20 0.36
FYN P06241 1/20 0.36
PGR P06401 1/20 0.36
HSP90AA1 P07900 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
ADRA2A P08913 1/20 0.36
CHRM1 P11229 1/20 0.36
TSHR P16473 1/20 0.36
ADRA2B P18089 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10843668 0.94 CYP3A4 (0.50) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL9834680 0.89 CYP3A4 (0.46) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL9833161 0.82 CYP3A4 (0.50) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL9833758 0.81 CYP3A4 (0.46) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL10845394 0.77 CYP3A4 (0.43) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL12095527 0.76 CYP3A4 (0.44) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL8815519 0.74 CYP3A4 (0.61) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL8815515 0.74 CYP3A4 (0.61) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL10505150 0.71 CYP3A4 (0.51) CYP3A4CYP2C9THRBCYP1A2CYP2D6
SCHEMBL9201668 0.70 CYP3A4 (0.62) CYP3A4CYP2C9THRBCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0133248-B1 1,2,4-TRIAZOL-1-YL-DERIVATIVES SHIONOGI & CO., LTD. (JP) 1991-11-21 EP claimed
EP-0133248-B1 1,2,4-TRIAZOL-1-YL-DERIVATIVES SHIONOGI & CO., LTD. (JP) 1991-11-21 EP disclosed
US-4612322-A FUNGICIDES SHIONOGI & CO., LTD. (JP) 1986-09-16 US disclosed
EP-0133248-A2 1,2,4-Triazol-1-yl-derivatives SHIONOGI & CO., LTD. (JP) 1985-02-20 EP disclosed