SCHEMBL983364

SCHEMBL983364

Cc1noc(-c2cccc(NC(=O)C(O)(CC3(c4ccccc4C(F)(F)F)CCC3)C(F)(F)F)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 16/20 0.44
KIF18A Q8NI77 1/20 0.42
TP53 P04637 2/20 0.41
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL985083 0.91 NR3C1 (0.44) NR3C1
SCHEMBL984371 0.81 RHOA (0.42) NR3C1
SCHEMBL5644235 0.78 NR3C1 (0.69) NR3C1
SCHEMBL7167931 0.77 NR3C1 (0.67) NR3C1
SCHEMBL5644049 0.76 NR3C1 (0.68) NR3C1
SCHEMBL986328 0.76 NR3C1 (0.40) NR3C1POLB
SCHEMBL983367 0.75 TP53 (0.41) KIF18ATP53POLBMAPT
SCHEMBL5641362 0.75 NR3C1 (0.69) NR3C1
SCHEMBL983406 0.74 EPHX2 (0.38) NR3C1TP53
SCHEMBL7169251 0.72 NR3C1 (0.61) NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960351-B1 PROPIONAMIDE COMPOUNDS AS ANTIINFLAMMATORY AGENTS HOFFMANN LA ROCHE (CH) 2013-06-19 EP claimed
US-7868031-B2 Propionamide compounds as antiinflammatory agents ROCHE PALO ALTO LLC (US) 2011-01-11 US claimed
EP-1960351-A1 PROPIONAMIDE COMPOUNDS AS ANTIINFLAMMATORY AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2008-08-27 EP claimed
US-20070135500-A1 Propionamide compounds as antiinflammatory agents ROCHE PALO ALTO LLC 2007-06-14 US claimed
WO-2007065821-A1 PROPIONAMIDE COMPOUNDS AS ANTIINFLAMMATORY AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2007-06-14 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070135500-A1 Propionamide compounds as antiinflammatory agents PTGS1, PTGER1, PTGES3 NR3C1 707/4885KIF18A 4174/4885TP53 4411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.