SCHEMBL9834875

SCHEMBL9834875

COc1c(OCC(F)(F)C(F)(F)F)ccnc1CSc1nc2ccccc2[nH]1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.66
NPC1 O15118 8/20 0.66
CYP1A2 P05177 3/20 0.66
CYP2D6 P10635 3/20 0.66
CYP2C9 P11712 3/20 0.66
CYP2C19 P33261 3/20 0.66
CYP3A4 P08684 2/20 0.66
NOS3 P29474 1/20 0.51
NOS1 P29475 1/20 0.51
NOS2 P35228 1/20 0.51
SMN1; SMN2 Q16637 7/20 0.50
KMT2A Q03164 4/20 0.47
NFKB1 P19838 3/20 0.47
NFKB2 Q00653 3/20 0.47
RELA Q04206 3/20 0.47
MEN1 O00255 2/20 0.47
LMNA P02545 3/20 0.45
TP53 P04637 2/20 0.45
CYP2C8 P10632 2/20 0.45
CYP2E1 P05181 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836498 0.92 RAB9A (0.78) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL6440543 0.88 RAB9A (0.85) RAB9ANPC1CYP1A2CYP2D6CYP2C9
Water SCHEMBL6737292 0.87 RAB9A (0.83) RAB9ANPC1CYP1A2CYP2D6CYP2C9
Water SCHEMBL6737289 0.87 RAB9A (0.83) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9835266 0.87 CYP2D6 (0.52) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9835253 0.87 CYP1A2 (0.52) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9833507 0.86 SMN1; SMN2 (0.62) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL6377443 0.86 RAB9A (0.66) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9835001 0.86 RAB9A (0.59) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL6377287 0.85 RAB9A (0.62) RAB9ANPC1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4738975-A Pyridine derivatives, and use as anti-ulcer agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-04-19 US claimed
EP-0208452-B1 PYRIDINE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1991-09-18 EP disclosed
US-4738975-A Pyridine derivatives, and use as anti-ulcer agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-04-19 US disclosed
EP-0208452-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-01-14 EP disclosed