SCHEMBL9834982

SCHEMBL9834982

CCOC(=O)C1(C)C(=O)Nc2cc3c(cc21)NC(C(C)C)N3

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ADCY8 P40145 1/20 0.34
FGB P02675 1/20 0.33
MAPT P10636 3/20 0.33
BRD4 O60885 1/20 0.33
POLB P06746 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
AKR1B1 P15121 1/20 0.31
KCNT1 Q5JUK3 1/20 0.31
LMNA P02545 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833652 0.86 ALDH1A1 (0.36) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9833693 0.85 ALDH1A1 (0.36) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9835788 0.85 MAPT (0.36) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9832994 0.83 TP53 (0.34) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9834518 0.83 ALDH1A1 (0.36) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9834073 0.82 ALDH1A1 (0.34) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9833426 0.81 MAPT (0.34) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9834678 0.81 TP53 (0.33) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9835044 0.80 SMN1; SMN2 (0.41) ALDH1A1TP53CYP1A2CYP2C9TSHR
SCHEMBL9832763 0.80 POLB (0.41) ALDH1A1TP53CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed