SCHEMBL9835112

SCHEMBL9835112

Cc1cnc(N2C(=O)c3ccccc3C2=O)c(C(Cl)Cl)n1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.38
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
HTT P42858 1/20 0.36
AR P10275 1/20 0.36
RXFP1 Q9HBX9 2/20 0.36
ALDH1A1 P00352 2/20 0.36
DPP4 P27487 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
GAA P10253 1/20 0.35
TLR9 Q9NR96 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836486 0.84 HTT (0.37) CASP3KMT2AMEN1HTTAR
SCHEMBL9834526 0.81 HTT (0.36) CASP3KMT2AMEN1HTTAR
SCHEMBL9836183 0.80 HTT (0.35) CASP3KMT2AMEN1HTTAR
SCHEMBL9833927 0.80 HCRTR1 (0.44) CASP3KMT2AMEN1HTTAR
SCHEMBL9837203 0.77 RXFP1 (0.38) KMT2AMEN1HTTARRXFP1
SCHEMBL9833878 0.77 CASP3 (0.38) CASP3KMT2AMEN1HTTAR
SCHEMBL10731348 0.73 RXFP1 (0.38) KMT2AMEN1HTTARRXFP1
SCHEMBL10730941 0.69 HTT (0.37) CASP3KMT2AMEN1HTTAR
SCHEMBL9834075 0.69 RXFP1 (0.39) CASP3KMT2AMEN1HTTAR
SCHEMBL9835091 0.69 HTT (0.35) CASP3KMT2AMEN1HTTAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0175263-B1 2-AMINO-3-CHLOROMETHYL-5-(DICHLOROMETHYL)-PYRAZINES AND PROCESS FOR THEIR PREPARATION BASF Aktiengesellschaft (DE) 1991-06-05 EP disclosed
US-4692527-A 2-amino-3,5-di-(halomethyl)-pyrazines and their preparation BASF AKTIENGESELLSCHAFT (DE) 1987-09-08 US disclosed
EP-0175263-A2 2-Amino-3-chloromethyl-5-(dichloromethyl)-pyrazines and process for their preparation BASF Aktiengesellschaft (DE) 1986-03-26 EP disclosed