SCHEMBL9835146

SCHEMBL9835146

O=C(O)C1=Cc2sc(C(c3ccccc3)n3ccnc3)cc2CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 5/20 0.71
CYP19A1 P11511 4/20 0.47
CYP11B1 P15538 4/20 0.46
CYP11B2 P19099 4/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
CYP26A1 O43174 4/20 0.43
CYP17A1 P05093 2/20 0.43
MEN1 O00255 1/20 0.43
NR1I2 O75469 1/20 0.43
USP2 O75604 1/20 0.43
ABCB11 O95342 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PLA2G1B P04054 1/20 0.43
TP53 P04637 1/20 0.43
PGR P06401 1/20 0.43
HSP90AA1 P07900 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
IDO1 P14902 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL27264309 0.96 TBXAS1 (0.67) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
SCHEMBL10553258 0.92 TBXAS1 (0.61) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
Water SCHEMBL9837182 0.91 TBXAS1 (0.60) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
SCHEMBL9836059 0.89 TBXAS1 (0.58) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
SCHEMBL9835130 0.87 TBXAS1 (0.57) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
SCHEMBL9401646 0.84 TBXAS1 (0.53) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
SCHEMBL9401641 0.84 TBXAS1 (0.53) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
SCHEMBL9836166 0.83 TBXAS1 (1.00) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
Water SCHEMBL9836190 0.76 TBXAS1 (0.82) TBXAS1CYP19A1CYP11B1CYP11B2PDE3B
SCHEMBL9837224 0.74 TBXAS1 (0.43) TBXAS1CYP19A1CYP11B1CYP11B2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0240107-B1 THIANAPHTHENE DERIVATIVES, THEIR PRODUCTION AND USE Sankyo Company Limited (JP) 1991-08-21 EP claimed
US-4847272-A ANTICOAGULANTS SANKYO COMPANY LIMITED (JP) 1989-07-11 US claimed
EP-0240107-A1 Thianaphthene derivatives, their production and use Sankyo Company Limited (JP) 1987-10-07 EP claimed