SCHEMBL9835368

SCHEMBL9835368

O=c1c2[nH]cnc2n(-c2ccccc2)c(=O)n1-c1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.76
PDE4A P27815 9/20 0.68
PDE4B Q07343 9/20 0.68
PDE4C Q08493 9/20 0.68
PDE4D Q08499 9/20 0.68
KMT2A Q03164 3/20 0.68
POLB P06746 2/20 0.57
MEN1 O00255 1/20 0.53
NPC1 O15118 1/20 0.50
ADORA3 P0DMS8 1/20 0.48
ADORA2B P29275 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9584926 0.86 MAPK1 (1.00) MAPK1PDE4APDE4BPDE4CPDE4D
SCHEMBL5964701 0.86 PDE4A (0.73) MAPK1PDE4APDE4BPDE4CPDE4D
SCHEMBL12013393 0.84 MAPK1 (0.56) MAPK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6662589 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL6244272 0.79 PDE4A (0.68) MAPK1PDE4APDE4BPDE4CPDE4D
SCHEMBL6664629 0.78 PDE4A (0.86) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL6665761 0.78 PDE4A (0.74) MAPK1PDE4APDE4BPDE4CPDE4D
SCHEMBL3612101 0.78 ADORA2B (0.69) MAPK1PDE4APDE4BPDE4CPDE4D
SCHEMBL7604842 0.77 PDE4A (0.65) MAPK1PDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL6660919 0.77 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0454773-A1 NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS Bundgaard, Hans (DK) 1991-11-06 EP claimed
WO-1990008128-A1 NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS BUNDGAARD HANS (DK) 1990-07-26 WO claimed