SCHEMBL9835375

SCHEMBL9835375

CC(=O)C1(C)C(=O)Nc2cc3[nH]c(C4=CCCC4)nc3cc21

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
AURKA O14965 1/20 0.38
AURKB Q96GD4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835724 0.86 AURKA (0.37) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9832792 0.85 PDE3B (0.53) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9835819 0.82 PDE3B (0.52) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833577 0.78 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10566074 0.77 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9832264 0.77 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9835803 0.77 HSP90AA1 (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833047 0.76 ALDH1A1 (0.42) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10564794 0.76 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9835860 0.76 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed