SCHEMBL9835832

SCHEMBL9835832

O=C=Nc1c(F)cc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
ALDH1A1 P00352 2/20 0.32
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
RECQL P46063 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964625 0.90 GABRA1 (0.38) MAPK1TDP1GABRA1GABRB2TSHR
SCHEMBL1019709 0.85 MAPK1 (0.45) MAPK1TDP1GABRA1GABRB2ALDH1A1
SCHEMBL1952585 0.84 MAPK1 (0.38) MAPK1TDP1GABRA1GABRB2
SCHEMBL28565932 0.81 GABRA1 (0.36) MAPK1TDP1GABRA1GABRB2CYP3A4
SCHEMBL3388964 0.81 GABRA1 (0.32) MAPK1TDP1GABRA1GABRB2
SCHEMBL17648937 0.80 GABRA1 (0.33) GABRA1GABRB2ALDH1A1CYP3A4TSHR
SCHEMBL28565654 0.78 KDM4E (0.38) MAPK1TDP1GABRA1GABRB2ALDH1A1
SCHEMBL10611282 0.78 GABRA1 (0.50) MAPK1TDP1GABRA1GABRB2
SCHEMBL28912552 0.78 MAPK1 (0.34) MAPK1TDP1GABRA1GABRB2
SCHEMBL1950823 0.77 MAPK1 (0.42) MAPK1TDP1GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248506-A Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-08-13 CN disclosed
CN-107001372-B Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-04-27 CN disclosed
EP-0241559-B1 OXAZOLIDINEDIONE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND HERBICIDES CONTAINING THE SAME SAGAMI CHEMICAL RESEARCH CENTER (JP) 1991-10-30 EP disclosed
US-4983751-A Chemical intermediates SAGAMI CHEMICAL RESEARCH CENTER (JP) 1991-01-08 US disclosed
US-4818272-A NONPHYTOTOXICITY FOR CROPS HELICAL STREAMS SAGAMI CHEMICAL RESEARCH CENTER (JP) 1989-04-04 US disclosed
EP-0241559-A1 OXAZOLIDINEDIONE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND HERBICIDES CONTAINING THE SAME SAGAMI CHEMICAL RESEARCH CENTER (JP) 1987-10-21 EP disclosed