SCHEMBL9835879

SCHEMBL9835879

Cc1ccc2c(c1)-c1c(c(C(=O)CC#N)nn1-c1ccccc1)CO2

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
PIK3CD O00329 2/20 0.44
PIK3R2 O00459 2/20 0.44
PIK3CA P42336 2/20 0.44
PIK3CB P42338 2/20 0.44
PIK3CG P48736 2/20 0.44
PIK3R5 Q8WYR1 2/20 0.44
PIK3R3 Q92569 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
MAPT P10636 3/20 0.39
TP53 P04637 6/20 0.38
NR1H4 Q96RI1 4/20 0.38
CCNA2 P20248 3/20 0.38
CDK2 P24941 3/20 0.38
CCNA1 P78396 3/20 0.38
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9834213 0.88 NR1H4 (0.47) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9834058 0.88 PTGS1 (0.43) ALDH1A1PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9833914 0.88 PTGS1 (0.44) ALDH1A1PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9831535 0.88 PIK3CD (0.46) ALDH1A1PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9832563 0.85 CCNA2 (0.37) ALDH1A1PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9523571 0.82 PIK3CD (0.54) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9835538 0.80 MAPT (0.51) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL9832768 0.80 CCNA2 (0.44) ALDH1A1PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9833312 0.80 ALDH1A1 (0.40) ALDH1A1PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9833649 0.80 PTGS1 (0.46) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed