SCHEMBL9835977

SCHEMBL9835977

O=C(O)/C=C/c1ccc(Oc2cccc(F)c2)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RHOA P61586 1/20 0.53
ALDH1A1 P00352 4/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
POLB P06746 1/20 0.48
KDM4E B2RXH2 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
P4HTM Q9NXG6 1/20 0.46
PKM P14618 1/20 0.45
KMT2A Q03164 2/20 0.45
RAB9A P51151 2/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
FFAR1 O14842 1/20 0.45
GSK3B P49841 1/20 0.44
BACE1 P56817 1/20 0.44
HRH3 Q9Y5N1 2/20 0.44
AKR1C3 P42330 3/20 0.43
MEN1 O00255 1/20 0.43
KCNH2 Q12809 1/20 0.43
EGLN1 Q9GZT9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835980 1.00 RHOA (0.53) RHOAALDH1A1L3MBTL1POLBKDM4E
SCHEMBL3179354 0.85 SRD5A2 (0.56) RHOAALDH1A1L3MBTL1KDM4ESMN1; SMN2
SCHEMBL3179345 0.85 SRD5A2 (0.56) RHOAALDH1A1L3MBTL1KDM4ESMN1; SMN2
SCHEMBL10666158 0.84 ALDH1A1 (0.70) RHOAALDH1A1L3MBTL1POLBKDM4E
SCHEMBL10666146 0.84 ALDH1A1 (0.70) RHOAALDH1A1L3MBTL1POLBKDM4E
SCHEMBL3618167 0.84 ALDH1A1 (0.65) ALDH1A1L3MBTL1KDM4ESMN1; SMN2P4HTM
SCHEMBL3618165 0.84 ALDH1A1 (0.65) ALDH1A1L3MBTL1KDM4ESMN1; SMN2P4HTM
SCHEMBL510406 0.81 ALDH1A1 (0.69) ALDH1A1L3MBTL1POLBKDM4EKMT2A
SCHEMBL28893686 0.80 KDM4E (0.58) RHOAALDH1A1POLBKDM4ESMN1; SMN2
SCHEMBL28893595 0.80 KDM4E (0.58) RHOAALDH1A1POLBKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0210782-B1 PYRIDINE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Dainippon Pharmaceutical Co., Ltd. (JP) 1991-04-17 EP disclosed
US-4778796-A ω-(3-pyridyl)alkenamide derivatives and anti-allergenic pharmaceutical compositions containing same DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1988-10-18 US disclosed
EP-0210782-A2 Pyridine compounds, process for the preparation thereof and pharmaceutical composition containing the same Dainippon Pharmaceutical Co., Ltd. (JP) 1987-02-04 EP disclosed