SCHEMBL9836258

SCHEMBL9836258

C=CC(=O)NC(C)(c1ccccc1)S(C)(=O)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
TGM2 P21980 6/20 0.46
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
EGFR P00533 2/20 0.37
NR3C2 P08235 1/20 0.37
PTPN1 P18031 1/20 0.36
PTPN11 Q06124 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28264187 0.88 CYP2C19 (0.51) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL5396951 0.78 ALDH1A1 (0.58) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL10594826 0.76 CYP2C19 (0.59) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL30758297 0.76 CYP2C19 (0.59) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL3701045 0.75 CYP2C19 (0.51) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL730210 0.74 ALDH1A1 (0.53) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL6908098 0.74 ALDH1A1 (0.53) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL10635375 0.74 CYP2C19 (0.50) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
SCHEMBL10534963 0.74 CYP2C19 (0.50) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2
Potassium Ion SCHEMBL9616863 0.74 CYP2C19 (0.50) ALDH1A1CYP3A4CYP2C9CYP2C19TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0272684-B1 DERIVATIVES OF N-(METHYLSULPHONYLPHENYLETHYL)-2-PROPENAMIDES AND THEIR USE AS ANTIBIOTICS ZAMBON S.p.A. (IT) 1991-06-12 EP disclosed
EP-0272684-A2 Derivatives of N-(methylsulphonylphenylethyl)-2-propenamides and their use as antibiotics ZAMBON S.p.A. (IT) 1988-06-29 EP disclosed