SCHEMBL9837622

SCHEMBL9837622

Nc1c(F)c(N2CCNCC2)c(Cl)c2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.61
KCNH2 Q12809 2/20 0.61
CACNA1F O60840 1/20 0.61
MAPK1 P28482 1/20 0.61
CACNA1D Q01668 1/20 0.61
CACNA1S Q13698 1/20 0.61
CACNA1C Q13936 1/20 0.61
GSK3B P49841 13/20 0.53
TOP2A P11388 2/20 0.51
TOP2B Q02880 2/20 0.51
ALDH1A1 P00352 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CHRM2 P08172 1/20 0.50
CHRM1 P11229 1/20 0.50
OPRM1 P35372 1/20 0.50
OPRD1 P41143 1/20 0.50
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6305453 0.91 KCNH2 (0.73) POLBKCNH2CACNA1FMAPK1CACNA1D
Hydrochloric Acid SCHEMBL10543998 0.90 KCNH2 (0.72) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL9167285 0.90 POLB (0.57) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL8437298 0.88 KCNH2 (0.64) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL8557613 0.88 KCNH2 (0.55) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL9837378 0.88 POLB (0.61) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL9837304 0.88 KCNH2 (0.69) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL10547807 0.87 KCNH2 (0.68) POLBKCNH2CACNA1FMAPK1CACNA1D
Hydrochloric Acid SCHEMBL9022804 0.87 KCNH2 (0.63) POLBKCNH2CACNA1FMAPK1CACNA1D
SCHEMBL9077977 0.86 POLB (0.55) POLBKCNH2CACNA1FMAPK1CACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0226961-B1 5-AMINO AND 5-HYDROXY-6,8-DIFLUOROQUINOLONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
US-4977154-A 7-PIPERAZINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1990-12-11 US claimed
EP-0226961-A1 5-Amino and 5-hydroxy-6,8-difluoroquinolones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1987-07-01 EP claimed
EP-0226961-B1 5-AMINO AND 5-HYDROXY-6,8-DIFLUOROQUINOLONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4977154-A 7-PIPERAZINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1990-12-11 US disclosed
EP-0226961-A1 5-Amino and 5-hydroxy-6,8-difluoroquinolones as antibacterial agents WARNER-LAMBERT COMPANY (US) 1987-07-01 EP disclosed