SCHEMBL9837945

SCHEMBL9837945

C=C1COc2c(N3CCC(N)C3)c(F)cc3c(=O)c4c(=O)[nH]oc4n1c23

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 15/20 0.41
TOP2B Q02880 10/20 0.41
TOP1 P11387 4/20 0.40
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
PIM1 P11309 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
PIM3 Q86V86 1/20 0.38
CSNK1G1 Q9HCP0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9839667 0.99 TOP2A (0.40) TOP2ATOP2BTOP1ALDH1A1POLB
SCHEMBL9839307 0.85 AADAT (0.33) ALDH1A1POLB
SCHEMBL9837703 0.85 KDM4E (0.42) ALDH1A1POLBOPRM1
SCHEMBL9839117 0.84 TOP2A (0.40) TOP2ATOP2BTOP1ALDH1A1POLB
SCHEMBL10729692 0.84 TOP2A (0.37) TOP2ATOP2BTOP1ALDH1A1POLB
Hydrochloric Acid SCHEMBL9839687 0.83 TOP2A (0.39) TOP2ATOP2BTOP1ALDH1A1POLB
SCHEMBL9839234 0.83 KDM4E (0.44) TOP2ATOP1ALDH1A1POLB
SCHEMBL9837629 0.82 PIM1 (0.45) TOP2ATOP2BTOP1ALDH1A1POLB
Hydrochloric Acid SCHEMBL9839219 0.81 PIM1 (0.44) TOP2ATOP2BTOP1ALDH1A1POLB
SCHEMBL9825021 0.79 PIM1 (0.43) TOP2ATOP2BTOP1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0228661-B1 ISOXAZOLO-PYRIDO-BENZOXAZINE AND ISOTHIAZOLO-PYRIDO-BENZOXAZINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4687770-A Isoxazolo-pyrido-benzoxazine and isothiazolo-pyrido-benzoxazine derivatives ABBOTT LABORATORIES (US) 1987-08-18 US disclosed
EP-0228661-A1 Isoxazolo-pyrido-benzoxazine and isothiazolo-pyrido-benzoxazine derivatives ABBOTT LABORATORIES (US) 1987-07-15 EP disclosed