SCHEMBL9838764

SCHEMBL9838764

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CC4CCC3CN4C)c(F)c21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.59
ALDH1A1 P00352 5/20 0.59
HPGD P15428 4/20 0.59
HSD17B10 Q99714 4/20 0.59
PMP22 Q01453 1/20 0.58
KCNH2 Q12809 5/20 0.48
DRD3 P35462 1/20 0.46
POLB P06746 2/20 0.44
OPRM1 P35372 2/20 0.44
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
OPRD1 P41143 1/20 0.44
TOP2A P11388 4/20 0.43
TOP2B Q02880 4/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
PRKD3 O94806 1/20 0.43
ALOX15 P16050 1/20 0.43
CLK2 P49760 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866403 0.96 KDM4E (0.58) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9838719 0.92 KDM4E (0.59) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9669484 0.87 TOP2A (0.58) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL9837294 0.85 KDM4E (0.64) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9837357 0.85 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9867237 0.84 TOP2A (0.55) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL9837564 0.84 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749429 0.84 KDM4E (0.67) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9838745 0.83 KDM4E (0.56) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749610 0.82 DRD3 (0.63) KDM4EALDH1A1HPGDHSD17B10DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0159174-B1 SUBSTITUTED NAPHTHYRIDINE-, QUINOLINE- AND BENZOXAZINE- CARBOXYLIC ACIDS AS ANTIBACTERIAL AGENTS AND PROCESSES FOR THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1991-10-23 EP disclosed
US-4571396-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1986-02-18 US disclosed
EP-0159174-A2 Substituted naphthyridine-, quinoline- and benzoxazine- carboxylic acids as antibacterial agents and processes for their production WARNER-LAMBERT COMPANY (US) 1985-10-23 EP disclosed