SCHEMBL9866403

SCHEMBL9866403

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CC4CCCC3CN4C)c(F)c21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.58
ALDH1A1 P00352 5/20 0.58
HPGD P15428 4/20 0.58
HSD17B10 Q99714 4/20 0.58
PMP22 Q01453 1/20 0.57
KCNH2 Q12809 4/20 0.45
DRD3 P35462 1/20 0.44
LMNA P02545 3/20 0.41
BRD4 O60885 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
CYP2J2 P51589 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
OPRM1 P35372 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9838764 0.96 KDM4E (0.59) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9838719 0.90 KDM4E (0.59) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9867237 0.87 TOP2A (0.55) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL9866672 0.85 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9837357 0.83 KDM4E (0.60) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9669484 0.83 TOP2A (0.58) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL9837564 0.83 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9837294 0.82 KDM4E (0.64) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9838745 0.81 KDM4E (0.56) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL10883769 0.81 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP claimed
US-4992546-A Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives WARNER-LAMBERT COMPANY (US) 1991-02-12 US disclosed
US-4968799-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1990-11-06 US disclosed
US-4962108-A A QUIN-4-ONE HAVING THE FOLLOWING RING SUBSTITUENTS; 1-ALKYL OR PHENYL, 3-CARBOXY DERIVATIVE, 6-FLUORO AND 8-BRIDGED N-HETEROCYCLIC RING WARNER-LAMBERT COMPANY (US) 1990-10-09 US disclosed
US-4923879-A CARBOXYLIC ACID DERIVATIVES WITH BRIDGED SIDECHAINS WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP disclosed