SCHEMBL9839019

SCHEMBL9839019

CCC(=O)OC(CC)c1nc2c(C(F)(F)F)cccc2c(O)c1C(=O)Nc1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
LMNA P02545 3/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 2/20 0.41
USP2 O75604 1/20 0.41
HTT P42858 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
AURKA O14965 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
PRKX P51817 1/20 0.37
PRKG1 Q13976 1/20 0.37
MAPKAPK5 Q8IW41 1/20 0.37
SRPK1 Q96SB4 1/20 0.37
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9839145 0.89 NPC1 (0.40) NPC1RAB9AALDH1A1KDM4ELMNA
SCHEMBL9838903 0.85 RAB9A (0.40) NPC1RAB9ALMNAMAPTHTT
SCHEMBL10664235 0.83 NPC1 (0.47) NPC1RAB9AALDH1A1KDM4ELMNA
SCHEMBL10946310 0.83 NPC1 (0.47) NPC1RAB9AALDH1A1KDM4ELMNA
SCHEMBL9839093 0.81 NPC1 (0.42) NPC1RAB9AALDH1A1KDM4ELMNA
SCHEMBL9838204 0.80 KDM4E (0.43) NPC1RAB9AALDH1A1KDM4ELMNA
SCHEMBL10518993 0.79 NPC1 (0.40) NPC1RAB9ALMNAHTTSMN1; SMN2
SCHEMBL10524820 0.79 HSPA5 (0.40) NPC1RAB9ALMNAHTTMEN1
SCHEMBL11370104 0.79 NPC1 (0.50) NPC1RAB9AALDH1A1KDM4ELMNA
SCHEMBL9605284 0.78 RAB9A (0.39) NPC1RAB9AKDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988708-A 3-Carbamoyl-4-hydroxy-2-carboxylmethyl quinoline analgesics, antiinflammatory agents ROUSSEL UCLAF (FR) 1991-01-29 US disclosed
US-4845105-A 4-OH-quinoline carboxylic acid amides having analgesic and anti-inflammatory activity ROUSSEL UCLAF (FR) 1989-07-04 US disclosed
US-4735951-A Novel 4-hydroxy-3-quinoline-carboxylates having analgesic and anti-inflammatory activity ROUSSEL UCLAF (FR) 1988-04-05 US disclosed