SCHEMBL9842840

SCHEMBL9842840

CCn1cnc2c1c(=O)n(CC(C)=O)c(=O)n2C1CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.53
PDE4A P27815 5/20 0.51
PDE4B Q07343 4/20 0.51
PDE4C Q08493 4/20 0.51
PDE4D Q08499 4/20 0.51
ADORA2B P29275 3/20 0.51
ADORA2A P29274 2/20 0.51
KMT2A Q03164 3/20 0.46
LMNA P02545 1/20 0.42
ESR1 P03372 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.42
NFKB1 P19838 1/20 0.42
ACHE P22303 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
EEF2K O00418 1/20 0.42
EEF2 P13639 1/20 0.42
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9842799 0.91 PDE4A (0.57) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842761 0.88 PDE4A (0.51) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842846 0.86 PDE4A (0.57) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842873 0.86 PDE4A (0.64) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842777 0.85 PDE4A (0.62) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842620 0.85 ADORA2B (0.68) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842890 0.84 PDE4A (0.75) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842797 0.84 PDE4A (0.71) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842854 0.84 PDE4A (0.57) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL9842849 0.83 PDE4A (0.70) TRPA1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0430025-A2 Xanthine compound, method for preparing thereof, and a pharmaceutical composition comprising the same HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1991-06-05 EP disclosed