SCHEMBL9842978

SCHEMBL9842978

CCCCCCc1cc2c(cc1C#Cc1cnc(CCCCC(=O)O)cn1)C(C)(C)CC(C)(C)S2

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.34
SCD O00767 1/20 0.33
LTB4R Q15722 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9843104 0.93 PPARA (0.32) PPARA
SCHEMBL8875595 0.92 PTGDR2 (0.35) PTGDR2
SCHEMBL8864984 0.90 CYP3A4 (0.33) PTGDR2
SCHEMBL9843011 0.87 PPARA (0.38) PPARAPTGDR2SCDLTB4R
SCHEMBL8865035 0.85 CYP3A4 (0.34) PTGDR2
SCHEMBL9843179 0.85 PPARA (0.35) PPARAPTGDR2SCD
SCHEMBL9530961 0.84 PPARA (0.39) PPARAPTGDR2SCDLTB4R
SCHEMBL8865411 0.83 CYP3A4 (0.35)
SCHEMBL8877174 0.82 ALDH1A1 (0.35) PTGDR2
SCHEMBL9843001 0.82 CYP3A4 (0.44) PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0419130-A2 Acetylenes disubstituted with a heteroaromatic group and A 2-substituted chromanyl, thiochromanyl or 1,2,3,4- tetrahydroquinolinyl group having retinoid-like activity ALLERGAN, INC. (US) 1991-03-27 EP disclosed