SCHEMBL9844937

SCHEMBL9844937

COC(=O)c1ccc(/C=C/c2cn(C)c3ncnc(N)c23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.41
RET P07949 4/20 0.40
ALDH1A1 P00352 3/20 0.39
EP300 Q09472 2/20 0.39
TP53 P04637 1/20 0.39
EGFR P00533 1/20 0.38
SRC P12931 1/20 0.38
KDR P35968 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 1/20 0.38
RPS6KA3 P51812 1/20 0.38
MAPT P10636 3/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 2/20 0.36
GLA P06280 1/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844938 1.00 PTPN1 (0.41) PTPN1RETALDH1A1EP300TP53
SCHEMBL22677981 0.79 SRC (0.55) EGFRSRCKDR
SCHEMBL29407781 0.79 SRC (0.55) EGFRSRCKDR
SCHEMBL13004526 0.79 RPS6KA3 (0.51) RETALDH1A1TP53SRCRPS6KA3
SCHEMBL9844770 0.76 EP300 (0.49) RETALDH1A1EP300TP53EGFR
SCHEMBL9844771 0.76 NPC1 (0.43) ALDH1A1TP53NPC1RAB9AMAPT
SCHEMBL14114544 0.74 MAP3K7 (0.39) RETEGFRSRCKDRRPS6KA3
SCHEMBL13004542 0.74 MAP3K7 (0.41) RPS6KA3
SCHEMBL16939051 0.73 EIF2AK3 (0.36) RETEGFRSRCKDR
SCHEMBL16939048 0.72 ADORA2A (0.41) RETEGFRSRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed