SCHEMBL9845277

SCHEMBL9845277

ClCOCC(COCc1ccccc1)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
CA1 P00915 4/20 0.46
CA2 P00918 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
TACR1 P25103 5/20 0.45
MAPK1 P28482 1/20 0.41
SLC1A1 P43005 1/20 0.40
KMT2A Q03164 1/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10581265 1.00 TSHR (0.48) TSHRCA1CA2CA7CA9
SCHEMBL4535810 0.91 TSHR (0.58) TSHRCA1CA2CA7CA9
SCHEMBL4088276 0.89 TSHR (0.52) TSHRCA1CA2CA7CA9
SCHEMBL9575753 0.85 TSHR (0.52) TSHRCA1CA2CA7CA9
SCHEMBL14125272 0.82 TSHR (0.48) TSHRCA1CA2CA7CA9
SCHEMBL6840474 0.82 TSHR (0.48) TSHRCA1CA2CA7CA9
SCHEMBL9575541 0.81 TSHR (0.56) TSHRCA1CA2CA7CA9
SCHEMBL19068463 0.81 CA1 (0.49) TSHRCA1CA2CA7CA9
SCHEMBL14814507 0.80 TSHR (0.50) TSHRCA1CA2CA7CA9
SCHEMBL828589 0.80 CA1 (0.51) TSHRCA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0452680-A1 Substituted purines, process for their preparation and their use as antiviral agents HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-23 EP disclosed
US-4880820-A VIRICIDES, HERPES VIRUS MERCK & CO., INC. (US) 1989-11-14 US disclosed
US-4801710-A Regioselective synthesis of 9-substituted purine acyclonucleoside derivatives MERCK & CO., INC. (US) 1989-01-31 US disclosed
EP-0130126-B1 (S)-9-(2,3-DIHYDROXY-1-PROPOXYMETHYL) GUANINE AND ITS ACYL DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS ANTIHERPETIC AGENTS MERCK & CO. INC. (US) 1987-08-26 EP disclosed
EP-0130126-A1 (S)-9-(2,3-dihydroxy-1-propoxymethyl) guanine and its acyl derivatives, their preparation and their application as antiherpetic agents MERCK & CO. INC. (US) 1985-01-02 EP disclosed