SCHEMBL9845496

SCHEMBL9845496

CN(C)C(=O)/C=C/C(=O)N1CC(C)(C)Oc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.35
FGFR4 P22455 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
GFER P55789 1/20 0.33
ALDH1A1 P00352 3/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 2/20 0.33
RAB9A P51151 1/20 0.33
APAF1 O14727 1/20 0.32
CACNA1B Q00975 1/20 0.32
APBA1 Q02410 1/20 0.32
MCL1 Q07820 1/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
DRD1 P21728 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9845497 1.00 AKR1B1 (0.40) AKR1B1L3MBTL1FGFR4KMT2AMEN1
SCHEMBL4971376 0.88 AKR1B1 (0.44) AKR1B1L3MBTL1FGFR4KMT2AMEN1
SCHEMBL4971386 0.88 AKR1B1 (0.44) AKR1B1L3MBTL1FGFR4KMT2AMEN1
SCHEMBL9142159 0.83 KMT2A (0.45) AKR1B1KMT2AMEN1ALDH1A1MAPT
SCHEMBL9142156 0.83 KMT2A (0.45) AKR1B1KMT2AMEN1ALDH1A1MAPT
SCHEMBL16101298 0.83 AKR1B1 (0.46) AKR1B1L3MBTL1FGFR4KMT2AMEN1
SCHEMBL450748 0.81 AKR1B1 (0.46) AKR1B1L3MBTL1KMT2AMEN1GFER
SCHEMBL9148051 0.77 AKR1B1 (0.46) AKR1B1L3MBTL1KMT2AMEN1GFER
SCHEMBL9147726 0.77 AKR1B1 (0.43) AKR1B1L3MBTL1KMT2AMEN1GFER
SCHEMBL446546 0.75 MAPT (0.45) AKR1B1ALDH1A1MAPTRAB9ARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432893-A2 Benzoxazine derivatives, their preparation and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-06-19 EP disclosed